摘要
以溴化亚铜作催化剂,DMF作溶剂,用N-(o-alkynylphenyl)imines亚胺在温和条件下环合-加成反应,一步合成吲哚衍生物,结果发现恶唑类吲哚在不同催化剂、不同底物种类及反应条件下的反应速度和产率具有较大差异性.
Using cuprous bromide as catalyst, DMF as solvent, indole derivatives are get from N-(o-alkynylphenyl)imines by one step cyclization-addition reaction under mild conditions. Results show that the reaction rate and yield of oxazolidinone indole have great differences under different catalysts, substrate types and reaction conditions.
出处
《新乡学院学报》
2012年第4期319-321,共3页
Journal of Xinxiang University
关键词
吲哚
串联反应
恶唑
indole
tandem reaction
oxazole