摘要
以2,4-二乙酰基间苯三酚为基础,通过改变一个酰基碳链的长度,合成了三个间苯三酚乙酰基衍生物,目标化合物经LC-MS进行了确证,室内生测试验结果表明,2-乙酰基-4-丙酰基间苯三酚与2-乙酰基-4-丁酰基间苯三酚对立枯丝核菌、禾谷丝核菌、灰葡萄孢具有明显的抑制作用。
Three phloroglucinol acetylated derivatives were synthesized with 2,4-diacetylphloroglucinol as the basis structure.All the compounds synthesized were confirmed by LC-MS.The results of preliminary bioassay showed that two compounds of 2-acetyl-4-propionylphloroglucinol and 2-acetyl-4-butyrylphloroglucinol had obvious inhibitive effect on Rhizoctonia solani,Rhizoctonia cerealis,and Botrytis cinerea.
出处
《广州化工》
CAS
2011年第17期32-34,共3页
GuangZhou Chemical Industry
基金
国家"十二五"科技支撑计划项目
以天然产物为母体的绿色农药研究(No:2011BAE06B004-11)
山东省科技发展计划项目
以吡喃酮与辣椒碱为母体的绿色农药研究(No:2011GNC11101)
关键词
间苯三酚
合成
酰化
生物活性
phloroglucinol
acetylation
synthesis
biological activity
