Two compounds with strongly insecticidal and fungicidal activity, Kurarinone and Sophoraflavanone G , were isolated from Sophora flavescens Ait under the direction of bioassay, and comfirmed by UV, IR, MS and NMR. The...Two compounds with strongly insecticidal and fungicidal activity, Kurarinone and Sophoraflavanone G , were isolated from Sophora flavescens Ait under the direction of bioassay, and comfirmed by UV, IR, MS and NMR. The insecticidal activity of flavonoids from Sophora flavescens Ait was first reported here. The study of structure-activity relationship indicated that the methylation of 5-hydroxy on the phenyl ring would decrease the insecticidal and fungicidal activity of flavonoids.展开更多
Eight derivatives of 1,3-dimethyl-5-methylthio-4-phenylhydrazonocarboxyl pyrazole were synthesized from 1,3-dimethyl-5-methylthio-4-hydrazinocarboxyl pyrazole. All compounds synthesized were identified by 1H NMR and e...Eight derivatives of 1,3-dimethyl-5-methylthio-4-phenylhydrazonocarboxyl pyrazole were synthesized from 1,3-dimethyl-5-methylthio-4-hydrazinocarboxyl pyrazole. All compounds synthesized were identified by 1H NMR and elemental analysis. Some of them exhibited certain growth inhibition action to Phoma asparagi, Alternaria solani, Gibberella zeae, Physalospora piricola, Colletotrichum lagenarium as tested in vitro at dosage of 50 mg/L.展开更多
文摘Two compounds with strongly insecticidal and fungicidal activity, Kurarinone and Sophoraflavanone G , were isolated from Sophora flavescens Ait under the direction of bioassay, and comfirmed by UV, IR, MS and NMR. The insecticidal activity of flavonoids from Sophora flavescens Ait was first reported here. The study of structure-activity relationship indicated that the methylation of 5-hydroxy on the phenyl ring would decrease the insecticidal and fungicidal activity of flavonoids.
文摘Eight derivatives of 1,3-dimethyl-5-methylthio-4-phenylhydrazonocarboxyl pyrazole were synthesized from 1,3-dimethyl-5-methylthio-4-hydrazinocarboxyl pyrazole. All compounds synthesized were identified by 1H NMR and elemental analysis. Some of them exhibited certain growth inhibition action to Phoma asparagi, Alternaria solani, Gibberella zeae, Physalospora piricola, Colletotrichum lagenarium as tested in vitro at dosage of 50 mg/L.